SCHEMBL28699883

SCHEMBL28699883

OC1(O)CCOc2cc(Cl)ccc21

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 5/20 0.67
AKR1B1 P15121 3/20 0.40
AHR P35869 2/20 0.36
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CREBBP Q92793 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
PDK2 Q15119 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29414588 0.78 MAP3K14 (0.60) MAP3K14AKR1B1AHRALDH1A1GAA
SCHEMBL19285552 0.78 MAP3K14 (0.60) MAP3K14AKR1B1AHRALDH1A1GAA
SCHEMBL19284979 0.77 MAP3K14 (0.57) MAP3K14AKR1B1MAPTNPC1RAB9A
SCHEMBL28970256 0.76 MAP3K14 (0.57) MAP3K14AKR1B1ALDH1A1GAAMAPT
SCHEMBL28970233 0.76 MAP3K14 (0.57) MAP3K14AKR1B1ALDH1A1GAAMAPT
SCHEMBL23976814 0.76 MAP3K14 (0.57) MAP3K14AKR1B1ALDH1A1GAAMAPT
SCHEMBL23976493 0.74 MAP3K14 (0.55) MAP3K14AKR1B1ALDH1A1MAPTNPC1
SCHEMBL28807542 0.73 MAP3K14 (0.39) MAP3K14AKR1B1
SCHEMBL21930582 0.70 MAP3K14 (0.56) MAP3K14AKR1B1MAPTNPC1
SCHEMBL21930580 0.70 MAP3K14 (0.56) MAP3K14AKR1B1MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114096546-A Macrocyclic spirocyclic derivatives useful as MCL-1 inhibitors 詹森药业有限公司 2022-02-25 CN disclosed