SCHEMBL2870341

SCHEMBL2870341

Fc1cc(-c2c[nH]nn2)cc(Cl)c1Nc1nc2ccncc2c2cnccc12

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 12/20 0.49
CSNK2A1 P68400 8/20 0.44
CSNK2A2 P19784 3/20 0.41
CSNK2B P67870 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3502708 0.86 JAK2 (0.49) JAK2CSNK2A1CSNK2A2CSNK2B
SCHEMBL2862333 0.85 JAK2 (0.73) JAK2CSNK2A1
SCHEMBL3500457 0.77 JAK2 (0.71) JAK2
SCHEMBL2877188 0.69 JAK2 (0.68) JAK2CSNK2A1CSNK2A2CSNK2B
SCHEMBL2879082 0.66 JAK2 (0.46) JAK2CSNK2A1CSNK2A2CSNK2B
SCHEMBL3500922 0.66 JAK2 (0.88) JAK2
SCHEMBL2876749 0.66 JAK2 (0.60) JAK2CSNK2A1CSNK2A2CSNK2B
SCHEMBL2869677 0.66 JAK2 (1.00) JAK2CSNK2A1CSNK2A2CSNK2B
SCHEMBL30601032 0.65
SCHEMBL30544790 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200612-A1 INHIBITORS OF JANUS KINASES Merck Sharp & Dohme Corp. (US) 2010-06-30 EP claimed
WO-2009035575-A1 INHIBITORS OF JANUS KINASES MERCK & CO., INC. (US) 2009-03-19 WO claimed
EP-2200612-A1 INHIBITORS OF JANUS KINASES Merck Sharp & Dohme Corp. (US) 2010-06-30 EP disclosed
WO-2009035575-A1 INHIBITORS OF JANUS KINASES MERCK & CO., INC. (US) 2009-03-19 WO disclosed