SCHEMBL2870902

SCHEMBL2870902

Cc1cnc(F)cc1-c1cccc2cc(-c3ccnc(Cl)n3)sc12

nearest known ligand 0.34

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2927723 0.84 CA12 (0.30)
SCHEMBL2876823 0.84 CYP1A2 (0.32)
SCHEMBL594142 0.83 CA12 (0.30)
SCHEMBL2919757 0.83 BTK (0.32)
SCHEMBL27776244 0.80 MAPK14 (0.34) MAPK14
SCHEMBL388918 0.78 AAK1 (0.38)
SCHEMBL1336736 0.77 JAK2 (0.36)
SCHEMBL27886176 0.77 GCKR (0.30)
SCHEMBL595970 0.75 RAF1 (0.31) MAPK14
SCHEMBL392616 0.75 CYP19A1 (0.36) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101563342-B Imidazolidinonyl aminopyrimidine compounds for the treatment' of cancer LILLY CO ELI 2012-09-05 CN disclosed
CN-101679396-B Triazolylaminopyrimidine compounds LILLY CO ELI 2012-06-06 CN disclosed
CN-101568539-B Imidazolidinonyl aminopyrimidine compounds for the treatment of cancer LILLY CO ELI 2012-04-25 CN disclosed
EP-2125794-B1 IMIDAZOLIDINONYL AMINOPYRIMIDINE COMPOUNDS FOR THE TREATMENT OF CANCER LILLY CO ELI (US) 2010-10-20 EP disclosed
EP-2125793-B1 IMIDAZOLIDINONYL AMINOPYRIMIDINE COMPOUNDS FOR THE TREATMENT OF CANCER LILLY CO ELI (US) 2010-09-01 EP disclosed
CN-101679396-A Triazolylaminopyrimidine compounds LILLY CO ELI 2010-03-24 CN disclosed
CN-101568539-A Imidazolidinonyl aminopyrimidine compounds for the treatment of cancer LILLY CO ELI (US) 2009-10-28 CN disclosed
CN-101563342-A Imidazolidinonyl aminopyrimidine compounds for the treatment' of cancer LILLY CO ELI (US) 2009-10-21 CN disclosed