SCHEMBL28709369

SCHEMBL28709369

COC(=O)CNC(=O)c1cccc(Cl)c1C(=O)NCc1ccc2c(c1)OCO2

nearest known ligand 0.71

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH2 P05091 1/20 0.71
HPGD P15428 7/20 0.60
POLB P06746 2/20 0.57
PKM P14618 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
TSHR P16473 1/20 0.54
GHSR Q92847 1/20 0.54
LMNA P02545 1/20 0.54
MAPK1 P28482 1/20 0.54
MMP13 P45452 1/20 0.54
ALDH1A1 P00352 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
TP53 P04637 1/20 0.53
CRHBP P24387 1/20 0.53
RECQL P46063 1/20 0.53
CRHR2 Q13324 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28718762 0.92 ALDH2 (0.67) ALDH2HPGDPOLBPKMTDP1
SCHEMBL28722877 0.89 ALDH2 (0.76) ALDH2HPGDPOLBTDP1MEN1
SCHEMBL28722876 0.85 ALDH2 (0.72) ALDH2HPGDPOLBPKMTDP1
SCHEMBL28716509 0.84 ALDH2 (0.78) ALDH2HPGDPOLBTDP1MEN1
SCHEMBL28259740 0.84 ALDH2 (0.82) ALDH2HPGDPOLBTDP1MEN1
SCHEMBL503808 0.84 ALDH2 (1.00) ALDH2HPGDPOLBMEN1KMT2A
SCHEMBL28259432 0.83 ALDH2 (0.80) ALDH2HPGDPOLBMEN1KMT2A
SCHEMBL29493346 0.83 KMT2A (0.69) ALDH2HPGDPOLBMEN1KMT2A
SCHEMBL28709378 0.83 KMT2A (0.69) ALDH2HPGDPOLBMEN1KMT2A
SCHEMBL10107742 0.82 ALDH2 (0.77) ALDH2HPGDPOLBTDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114149386-A Aryl pentadiene amide aldehyde dehydrogenase inhibitor, and synthesis method and application thereof 中国人民解放军第二军医大学 2022-03-08 CN disclosed