SCHEMBL28752136

SCHEMBL28752136

CCN(C#N)c1ccccc1C(=O)Cn1c(=O)c2c(nc(N3CCCC(N)C3)n2CC=C(C)C)n(C)c1=O

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.72
CHRM1 P11229 2/20 0.72
CHRM2 P08172 1/20 0.72
CHRM3 P20309 1/20 0.72
KCNH2 Q12809 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28749934 0.93 DPP4 (0.74) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL556165 0.90 DPP4 (0.71) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL27583114 0.88 DPP4 (0.77) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL556290 0.88 DPP4 (0.74) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL556331 0.86 DPP4 (0.81) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL637179 0.86 DPP4 (0.81) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL555257 0.86 DPP4 (0.81) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL555776 0.86 DPP4 (0.81) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL637216 0.86 DPP4 (0.84) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL556657 0.86 DPP4 (0.73) DPP4CHRM1CHRM2CHRM3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101293888-B Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA 2013-09-25 CN disclosed
CN-101293888-A Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA (DE) 2008-10-29 CN disclosed
CN-100408579-C Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA (DE) 2008-08-06 CN disclosed
CN-1492870-A Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions ���ָ��Ӣ��ķ�������Ϲ�˾ 2004-04-28 CN disclosed