SCHEMBL28752138

SCHEMBL28752138

Cn1c(=O)n(CCc2ccccc2)c(=O)c2c1nc(N1CCCC(N)C1)n2CCc1ccccc1

nearest known ligand 0.82

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 19/20 0.82
CHRM1 P11229 5/20 0.64
CHRM3 P20309 2/20 0.64
CHRM2 P08172 1/20 0.64
KCNH2 Q12809 1/20 0.64
ALDH1A1 P00352 1/20 0.61
LMNA P02545 1/20 0.61
MAPT P10636 1/20 0.61
TSHR P16473 1/20 0.61
POU2F2 P09086 1/20 0.60
ADORA3 P0DMS8 1/20 0.60
POU2F1 P14859 1/20 0.60
HRH2 P25021 1/20 0.60
MC4R P32245 1/20 0.60
FAP Q12884 1/20 0.60
DPP8 Q6V1X1 1/20 0.60
DPP9 Q86TI2 1/20 0.60
GHSR Q92847 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL556428 0.96 DPP4 (0.82) DPP4CHRM1CHRM3CHRM2KCNH2
SCHEMBL555521 0.94 DPP4 (0.85) DPP4CHRM1CHRM3CHRM2KCNH2
SCHEMBL555576 0.94 DPP4 (0.76) DPP4CHRM1CHRM3CHRM2KCNH2
SCHEMBL27583065 0.92 DPP4 (0.75) DPP4CHRM1CHRM3CHRM2KCNH2
SCHEMBL556151 0.92 DPP4 (0.77) DPP4CHRM1CHRM3POU2F2ADORA3
SCHEMBL28346678 0.92 DPP4 (0.77) DPP4CHRM1CHRM3POU2F2ADORA3
SCHEMBL555833 0.90 DPP4 (1.00) DPP4CHRM1CHRM3CHRM2KCNH2
SCHEMBL4668687 0.90 DPP4 (0.71) DPP4
SCHEMBL555375 0.90 DPP4 (1.00) DPP4CHRM1CHRM3CHRM2KCNH2
SCHEMBL554218 0.90 DPP4 (1.00) DPP4CHRM1CHRM3CHRM2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101293888-B Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA 2013-09-25 CN disclosed
CN-101293888-A Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA (DE) 2008-10-29 CN disclosed
CN-100408579-C Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA (DE) 2008-08-06 CN disclosed
CN-1492870-A Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions ���ָ��Ӣ��ķ�������Ϲ�˾ 2004-04-28 CN disclosed