SCHEMBL28752829

SCHEMBL28752829

C=CC(c1ccc2c(c1)OC(c1ccc(F)cc1)(c1cccc(Cl)c1)O2)S(=O)(=O)N1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 14/20 0.43
GPR183 P32249 2/20 0.33
DRD5 P21918 1/20 0.33
SLC6A2 P23975 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRK1 P41145 1/20 0.33
HTR2B P41595 1/20 0.33
SLC6A3 Q01959 1/20 0.33
TMEM97 Q5BJF2 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
GPR35 Q9HC97 1/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GLRA3 O75311 1/20 0.31
GLRB P48167 1/20 0.31
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27625936 0.92 CNR1 (0.42) CNR1GPR183DRD5SLC6A2HTR2A
SCHEMBL27625938 0.91 CNR1 (0.53) CNR1OPRM1OPRK1KMT2AALDH1A1
SCHEMBL27607338 0.86 CNR1 (0.43) CNR1GPR183DRD5SLC6A2HTR2A
SCHEMBL28755841 0.81 CNR1 (0.45) CNR1GPR183DRD5SLC6A2HTR2A
SCHEMBL4476817 0.80 CNR1 (0.69) CNR1GPR183KMT2AMEN1ALDH1A1
SCHEMBL4464890 0.70 CNR1 (0.69) CNR1KMT2AMEN1ALDH1A1LMNA
SCHEMBL4466755 0.69 CNR1 (0.86) CNR1ALDH1A1LMNAMAPT
SCHEMBL4460616 0.69 CNR1 (0.77) CNR1ALDH1A1LMNAGAAMAPT
SCHEMBL1317004 0.67 CNR1 (0.64) CNR1GPR183DRD5SLC6A2HTR2A
SCHEMBL4461879 0.66 CNR1 (0.67) CNR1GPR183DRD5SLC6A2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100486973-C Novel benzodioxoles HOFFMANN LA ROCHE (CH) 2009-05-13 CN claimed
CN-1671684-A New benzodioxoles HOFFMANN LA ROCHE (CH) 2005-09-21 CN claimed
CN-100486973-C Novel benzodioxoles HOFFMANN LA ROCHE (CH) 2009-05-13 CN disclosed
CN-1671684-A New benzodioxoles HOFFMANN LA ROCHE (CH) 2005-09-21 CN disclosed