Acetic Acid

Acetic Acid

SCHEMBL28757239

CC(=O)O.O=C(Nc1cccc2[nH]ncc12)NC1CCc2cc(C(F)(F)F)ccc21

nearest known ligand 0.93

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Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Acetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 20/20 0.93
TRPV4 Q9HBA0 1/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1860664 0.96 TRPV1 (1.00) TRPV1TRPV4
Abt-102 SCHEMBL29388297 0.89 TRPV1 (1.00) TRPV1TRPV4
Abt-102 SCHEMBL29857846 0.89 TRPV1 (1.00) TRPV1TRPV4
Abt-102 SCHEMBL1854692 0.89 TRPV1 (1.00) TRPV1TRPV4
Abt-102 SCHEMBL1857275 0.89 TRPV1 (1.00) TRPV1TRPV4
Abt-102 SCHEMBL1859296 0.89 TRPV1 (1.00) TRPV1TRPV4
Acetic Acid SCHEMBL27762603 0.86 TRPV1 (0.93) TRPV1TRPV4
SCHEMBL1854750 0.86 TRPV1 (0.83) TRPV1TRPV4
SCHEMBL1859323 0.86 TRPV1 (0.83) TRPV1TRPV4
SCHEMBL1859424 0.86 TRPV1 (1.00) TRPV1TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102617464-A fused compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor ABBOTT LAB 2012-08-01 CN claimed
CN-1835924-A Fused compounds that inhibit vanilloid receptor subtype 1(vr1) receptor ABBOTT LAB (US) 2006-09-20 CN claimed
CN-1835924-A Fused compounds that inhibit vanilloid receptor subtype 1(vr1) receptor ABBOTT LAB (US) 2006-09-20 CN disclosed