SCHEMBL28758570

SCHEMBL28758570

CC(C)n1cc(-c2nc(C(=O)NCC[SnH](C)C)c(N)nc2-c2ccccc2)ccc1=O

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.47
ADORA1 P30542 5/20 0.44
ADORA2B P29275 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585113 0.89 ADORA2A (0.49) ADORA2AADORA1ADORA2B
SCHEMBL4584106 0.87 ADORA2A (0.47) ADORA2AADORA1ADORA2B
SCHEMBL4584042 0.85 ADORA2A (0.49) ADORA2AADORA1ADORA2B
SCHEMBL4584769 0.84 ADORA2A (0.47) ADORA2AADORA1ADORA2B
SCHEMBL4583361 0.83 ADORA2A (0.46) ADORA2AADORA1
SCHEMBL4584817 0.81 ADORA2A (0.51) ADORA2AADORA1
SCHEMBL4585347 0.81 ADORA2A (0.53) ADORA2AADORA1ADORA2B
SCHEMBL4585332 0.81 ADORA2A (0.48) ADORA2AADORA1
SCHEMBL4584074 0.81 ADORA2A (0.50) ADORA2AADORA1
SCHEMBL4584514 0.81 ADORA2A (0.50) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1871231-A Pyrazine derivatives and pharmaceutical use thereof ASTELLAS PHARMA INC (JP) 2006-11-29 CN disclosed