SCHEMBL28759231

SCHEMBL28759231

BrCCc1ccc2nc(-c3ccccc3)sc2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.59
SMN1; SMN2 Q16637 5/20 0.59
MAPT P10636 5/20 0.59
GLA P06280 4/20 0.59
GAA P10253 4/20 0.59
HPGD P15428 4/20 0.59
PKM P14618 3/20 0.59
ALDH1A1 P00352 2/20 0.59
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
NFKB1 P19838 3/20 0.56
NFKB2 Q00653 3/20 0.56
RELA Q04206 3/20 0.56
LMNA P02545 1/20 0.56
APP P05067 9/20 0.48
NPC1 O15118 6/20 0.47
RAB9A P51151 6/20 0.47
STAT1 P42224 1/20 0.47
TP53 P04637 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL506665 0.88 KDM4E (0.62) KDM4ESMN1; SMN2MAPTGLAGAA
SCHEMBL28265561 0.85 SMN1; SMN2 (0.59) KDM4ESMN1; SMN2MAPTGLAGAA
SCHEMBL27638532 0.84 S1PR1 (0.52) KDM4ESMN1; SMN2MAPTGLAGAA
SCHEMBL28265577 0.82 KDM4E (0.56) KDM4ESMN1; SMN2MAPTGLAGAA
SCHEMBL10230259 0.81 KDM4E (0.62) KDM4ESMN1; SMN2MAPTGLAGAA
SCHEMBL12967444 0.81 SMN1; SMN2 (0.62) KDM4ESMN1; SMN2MAPTGLAGAA
SCHEMBL507537 0.81 KDM4E (0.67) KDM4ESMN1; SMN2MAPTGLAGAA
SCHEMBL12596887 0.81 APP (0.68) KDM4ESMN1; SMN2MAPTGLAGAA
SCHEMBL12596888 0.81 KDM4E (0.62) KDM4ESMN1; SMN2MAPTGLAGAA
SCHEMBL27652217 0.79 TDP1 (0.42) KDM4ESMN1; SMN2MAPTGLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102329267-A 6-substituted 2,3,4, 5-tetrahydro-1H-benzo [d] aza as 5-HT2Creceptor agonists LILLY CO ELI 2012-01-25 CN disclosed
CN-102311387-A 6-substituted 2,3,4, 5-tetrahydro-1H-benzo [d] aza as 5-HT2Creceptor agonists LILLY CO ELI 2012-01-11 CN disclosed
CN-1934088-A As 5-HT2c6-substituted 2,3,4, 5-tetrahydro-1H-benzo [ d ] receptor agonists]Aza * LILLY CO ELI (US) 2007-03-21 CN disclosed