SCHEMBL28772016

SCHEMBL28772016

O=Cc1cc(Br)cc(OCc2ccc(Cl)cc2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 10/20 0.57
MAOA P21397 7/20 0.57
TACR2 P21452 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
TLR4 O00206 1/20 0.46
TLR2 O60603 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
LMNA P02545 1/20 0.45
APP P05067 1/20 0.44
NR4A2 P43354 2/20 0.43
CCR5 P51681 2/20 0.43
PLAT P00750 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29690200 1.00 MAOB (0.57) MAOBMAOATACR2L3MBTL1ALDH1A1
SCHEMBL31384354 0.89 TACR2 (0.55) MAOBMAOATACR2L3MBTL1ALDH1A1
SCHEMBL30823523 0.85 MAOB (0.65) MAOBMAOAALDH1A1CYP1A2TLR4
SCHEMBL16990010 0.85 MAOB (0.65) MAOBMAOAALDH1A1CYP1A2TLR4
SCHEMBL13321706 0.84 MAOB (0.55) MAOBMAOAAPPNR4A2CCR5
SCHEMBL3639311 0.84 NPC1 (0.66) MAOBMAOAALDH1A1TLR4TLR2
SCHEMBL18001687 0.79 MAOB (0.47) MAOBMAOATACR2L3MBTL1ALDH1A1
SCHEMBL18002178 0.79 MAOB (0.47) MAOBMAOATACR2L3MBTL1ALDH1A1
SCHEMBL18002505 0.79 MAOB (0.47) MAOBMAOATACR2L3MBTL1ALDH1A1
SCHEMBL8985612 0.79 MAOB (0.74) MAOBMAOATACR2TLR4TLR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114671815-B Aryl barbiturates compound and preparation method and application thereof 中国医学科学院药物研究所 2024-05-14 CN disclosed
CN-117430570-A Rhodamine acetic acid compound, and pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-01-23 CN disclosed
CN-114671815-A Aryl barbiturates compound and preparation method and application thereof 中国医学科学院药物研究所 2022-06-28 CN disclosed