SCHEMBL28778796

SCHEMBL28778796

COc1cccc(Cc2ccc(=O)[nH]n2)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALPL P05186 3/20 0.49
HTR1B P28222 1/20 0.47
CMA1 P23946 1/20 0.47
IDH1 O75874 2/20 0.46
CYP3A4 P08684 2/20 0.46
DAO P14920 1/20 0.46
TAAR1 Q96RJ0 2/20 0.45
CNR1 P21554 1/20 0.45
GPR55 Q9Y2T6 1/20 0.45
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44
VKORC1 Q9BQB6 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377193 0.84 CYP3A4 (0.50) CYP3A4DAOLMNA
SCHEMBL5369070 0.84 CYP3A4 (0.47) ALPLCYP3A4
SCHEMBL5413137 0.83 CYP3A4 (0.50) ALPLIDH1CYP3A4LMNA
SCHEMBL5373837 0.83 CYP3A4 (0.47) ALPLCYP3A4LMNA
SCHEMBL5376945 0.83 CYP3A4 (0.44) ALPLCYP3A4LMNA
SCHEMBL5376942 0.82 CYP3A4 (0.54) ALPLCYP3A4CNR1GPR55LMNA
SCHEMBL5374289 0.81 CYP3A4 (0.64) CYP3A4
SCHEMBL18127144 0.81 PTGS1 (0.51) CYP3A4DAOLMNA
SCHEMBL5377482 0.80 CYP3A4 (0.57) CYP3A4
SCHEMBL5367047 0.80 CYP3A4 (0.54) CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100469769-C Benzyl-pyridazinons as reverse transcriptase inhibitors ROCHE PALO ALTO LLC (CH) 2009-03-18 CN claimed