SCHEMBL28779558

SCHEMBL28779558

NC(=O)c1ccccc1-c1cc(-c2ccnc(N)n2)[nH]c1-c1ccccc1Cl

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 13/20 0.84
CDC7 O00311 11/20 0.66
CDK1 P06493 4/20 0.66
CDK2 P24941 4/20 0.66
GSK3B P49841 4/20 0.66
TAOK1 Q7L7X3 4/20 0.66
CDK9 P50750 3/20 0.66
PLK4 O00444 3/20 0.66
MAPK13 O15264 3/20 0.66
DAPK3 O43293 3/20 0.66
DYRK3 O43781 3/20 0.66
PRKD3 O94806 3/20 0.66
PRKCG P05129 3/20 0.66
PRKACA P17612 3/20 0.66
MARK3 P27448 3/20 0.66
MAPK1 P28482 3/20 0.66
FRK P42685 3/20 0.66
MAPK8 P45983 3/20 0.66
MAPK9 P45984 3/20 0.66
CSNK1A1 P48729 3/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27833178 0.99 JAK2 (0.82) JAK2CDC7CDK1CDK2GSK3B
SCHEMBL1208333 0.91 JAK2 (1.00) JAK2CDC7CDK1CDK2GSK3B
SCHEMBL28779568 0.91 JAK2 (0.70) JAK2CDC7CDK1CDK2GSK3B
SCHEMBL27738648 0.91 JAK2 (0.70) JAK2CDC7CDK1CDK2GSK3B
SCHEMBL27738546 0.91 JAK2 (0.70) JAK2CDC7CDK1CDK2GSK3B
Hydrochloric Acid SCHEMBL1133998 0.90 JAK2 (0.98) JAK2CDC7CDK1CDK2GSK3B
Hydrochloric Acid SCHEMBL28794392 0.90 JAK2 (0.68) JAK2CDC7CDK1CDK2GSK3B
SCHEMBL27759225 0.90 JAK2 (0.68) JAK2CDC7CDK1CDK2GSK3B
SCHEMBL28806454 0.88 JAK2 (0.65) JAK2CDC7CDK1CDK2GSK3B
SCHEMBL28779570 0.87 JAK2 (0.67) JAK2CDC7CDK1CDK2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101410387-A Pyridyl-and pyrimidinyl-substituted pyrrole-, thiophene-and furan-derivatives as kinase inhibitors NERVIANO MEDICAL SCIENCES SRL (IT) 2009-04-15 CN claimed
CN-102036983-A Process for the preparation of 5-(2-amino-pyrimidin-4-yl)-2-aryl-1h-pyrrole-3-carboxamides NERVIANO MEDICAL SCIENCES SRL 2011-04-27 CN disclosed
CN-101410387-A Pyridyl-and pyrimidinyl-substituted pyrrole-, thiophene-and furan-derivatives as kinase inhibitors NERVIANO MEDICAL SCIENCES SRL (IT) 2009-04-15 CN disclosed