SCHEMBL2878155

SCHEMBL2878155

COC(OC)c1c(-c2cccc3ccsc23)ccnc1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.31
DRD1 P21728 2/20 0.31
CYP2A6 P11509 1/20 0.31
ADRB2 P07550 1/20 0.31
CHRM2 P08172 1/20 0.31
ADRB1 P08588 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA2A P08913 1/20 0.31
CHRM1 P11229 1/20 0.31
DRD2 P14416 1/20 0.31
CHRM3 P20309 1/20 0.31
DRD4 P21917 1/20 0.31
DRD5 P21918 1/20 0.31
HRH2 P25021 1/20 0.31
HTR1D P28221 1/20 0.31
HTR1B P28222 1/20 0.31
HTR2A P28223 1/20 0.31
HTR1E P28566 1/20 0.31
HTR7 P34969 1/20 0.31
ADRA1A P35348 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2922383 0.76 ATR (0.38) SCN9ADRD1CYP2A6ADRB2CHRM2
SCHEMBL2878150 0.74
SCHEMBL2878488 0.72 CDK4 (0.32)
SCHEMBL391666 0.65 CYP2A6 (0.38) SCN9ADRD1CYP2A6ADRB2CHRM2
SCHEMBL391300 0.65 CACNA2D1 (0.34) SCN9AHTR2AATR
SCHEMBL1338523 0.64 ATR (0.35) SCN9ADRD1CYP2A6ADRB2CHRM2
SCHEMBL19756681 0.64 PDPK1 (0.46) CYP2A6ADRA1AHTR3AATR
SCHEMBL1339030 0.64 MAPT (0.30)
SCHEMBL14831141 0.63 CYP17A1 (0.43) SCN9ADRD1CYP2A6ATR
SCHEMBL594951 0.62 PRKCI (0.38) SCN9ACYP2A6ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125794-B1 IMIDAZOLIDINONYL AMINOPYRIMIDINE COMPOUNDS FOR THE TREATMENT OF CANCER LILLY CO ELI (US) 2010-10-20 EP disclosed