SCHEMBL28782016

SCHEMBL28782016

C=CC(NCCCC)S(=O)(=O)NC(=O)/C=C/c1c(C)nn(C)c1-n1ccc2cc(C#N)ccc21

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 2/20 0.31
FFAR4 Q5NUL3 1/20 0.31
NPY5R Q15761 1/20 0.31
HDAC1 Q13547 2/20 0.30
TBXA2R P21731 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27772611 0.90 HDAC1 (0.32) HDAC1
SCHEMBL27772816 0.89 HDAC1 (0.32) HDAC1
SCHEMBL27794146 0.89 PPARG (0.36) HDAC1
SCHEMBL27794135 0.87 TLR8 (0.34) HDAC1
SCHEMBL962196 0.87 CXCR2 (0.36) IRAK4FFAR4NPY5RHDAC1TBXA2R
SCHEMBL962198 0.87 CXCR2 (0.36) IRAK4FFAR4NPY5RHDAC1TBXA2R
SCHEMBL27772597 0.85 HDAC1 (0.32) HDAC1
SCHEMBL27772683 0.85 PPARG (0.36) HDAC1
SCHEMBL965770 0.84 PPARG (0.38) IRAK4FFAR4TBXA2R
SCHEMBL965767 0.84 PPARG (0.38) IRAK4FFAR4TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101646653-A Fused ring compounds as partial agonists of ppar-gamma TAKEDA PHARMACEUTICAL JP 2010-02-10 CN disclosed