SCHEMBL28786259

SCHEMBL28786259

CC(Nc1ncnc2[nH]cnc12)c1cc2ccc(F)cc2nc1-c1cccc(F)n1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 18/20 0.61
PIK3CG P48736 5/20 0.61
PIK3CA P42336 2/20 0.61
PIK3CB P42338 2/20 0.61
MAP4K4 O95819 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12005462 1.00 PIK3CD (0.61) PIK3CDPIK3CGPIK3CAPIK3CBMAP4K4
Amg-319 SCHEMBL16799298 0.89 PIK3CD (0.76) PIK3CDPIK3CGPIK3CAPIK3CB
Amg-319 SCHEMBL4185718 0.89 PIK3CD (0.76) PIK3CDPIK3CGPIK3CAPIK3CB
Amg-319 SCHEMBL17240940 0.88 PIK3CD (0.75) PIK3CDPIK3CGPIK3CAPIK3CB
SCHEMBL4171127 0.87 PIK3CD (0.57) PIK3CDPIK3CGPIK3CAPIK3CBMAP4K4
SCHEMBL27802785 0.87 PIK3CD (0.57) PIK3CDPIK3CGPIK3CAPIK3CBMAP4K4
SCHEMBL4174885 0.86 PIK3CD (0.59) PIK3CDPIK3CGPIK3CAPIK3CBMAP4K4
SCHEMBL4182647 0.86 PIK3CD (0.59) PIK3CDPIK3CGPIK3CAPIK3CBMAP4K4
SCHEMBL12005493 0.85 PIK3CD (0.56) PIK3CDPIK3CGPIK3CAPIK3CBMAP4K4
SCHEMBL10285587 0.84 PIK3CD (0.59) PIK3CDPIK3CGPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101715453-B Heterocyclic compounds and their uses AMGEN INC 2012-06-27 CN disclosed
CN-101715453-A Heterogeneous ring compound and application thereof AMGEN INC 2010-05-26 CN disclosed