SCHEMBL28789482

SCHEMBL28789482

Nc1ccccc1NC(=O)c1ccc(CNC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)c2ccccc2)cc1

nearest known ligand 0.84

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 13/20 0.84
HDAC3 O15379 12/20 0.84
HDAC2 Q92769 12/20 0.84
NCOR2 Q9Y618 4/20 0.84
TACR1 P25103 1/20 0.66
HDAC6 Q9UBN7 3/20 0.62
HDAC4 P56524 2/20 0.62
HDAC7 Q8WUI4 2/20 0.62
HDAC10 Q969S8 2/20 0.62
HDAC11 Q96DB2 2/20 0.62
HDAC8 Q9BY41 2/20 0.62
HDAC9 Q9UKV0 2/20 0.62
HDAC5 Q9UQL6 2/20 0.62
CTSL P07711 1/20 0.62
ERAP2 Q6P179 2/20 0.58
ERAP1 Q9NZ08 2/20 0.58
LNPEP Q9UIQ6 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27839978 0.92 HDAC1 (0.80) HDAC1HDAC3HDAC2NCOR2TACR1
SCHEMBL27839974 0.92 HDAC1 (0.80) HDAC1HDAC3HDAC2NCOR2TACR1
SCHEMBL27820625 0.88 HDAC1 (0.75) HDAC1HDAC3HDAC2NCOR2TACR1
SCHEMBL27839976 0.87 HDAC1 (0.70) HDAC1HDAC3HDAC2NCOR2HDAC6
SCHEMBL28793104 0.85 HDAC1 (0.70) HDAC1HDAC3HDAC2NCOR2TACR1
SCHEMBL28793141 0.84 HDAC1 (0.67) HDAC1HDAC3HDAC2NCOR2TACR1
SCHEMBL27820632 0.83 HDAC1 (0.67) HDAC1HDAC3HDAC2NCOR2TACR1
SCHEMBL27820613 0.83 HDAC1 (0.65) HDAC1HDAC3HDAC2NCOR2TACR1
SCHEMBL3557636 0.80 HDAC1 (0.62) HDAC1HDAC3HDAC2NCOR2HDAC6
SCHEMBL9271917 0.79 TACR1 (1.00) HDAC1HDAC3HDAC2NCOR2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102180826-A Histone deacetylase inhibitor containing alpha amino acid structure and application thereof UNIV CHINA PHARMA 2011-09-14 CN disclosed