SCHEMBL28790980

SCHEMBL28790980

Cc1ccc(C(=O)Nc2cccc(C(C)Nc3ncnc4ccc(Cl)cc34)c2)cn1

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 19/20 0.72
AURKA O14965 17/20 0.72
AURKB Q96GD4 3/20 0.67
CSF1R P07333 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL665542 0.85 RPS6KB1 (0.86) RPS6KB1AURKAAURKBCSF1R
SCHEMBL666838 0.84 RPS6KB1 (1.00) RPS6KB1AURKAAURKB
SCHEMBL665132 0.80 AURKA (1.00) RPS6KB1AURKAAURKB
SCHEMBL27830387 0.80 RPS6KB1 (0.76) RPS6KB1AURKAAURKB
SCHEMBL666018 0.80 AURKA (1.00) RPS6KB1AURKAAURKB
SCHEMBL27830109 0.77 RPS6KB1 (0.75) RPS6KB1AURKAAURKB
SCHEMBL3472939 0.75 CSF1R (1.00) RPS6KB1AURKAAURKBCSF1R
SCHEMBL29119483 0.75 CSF1R (1.00) RPS6KB1AURKAAURKBCSF1R
SCHEMBL30672123 0.75 CSF1R (1.00) RPS6KB1AURKAAURKBCSF1R
SCHEMBL667740 0.74 RPS6KB1 (0.83) RPS6KB1AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102317269-A Novel amino aza heterocyclic carboxamides MERCK PATENT GMBH 2012-01-11 CN disclosed