SCHEMBL28797161

SCHEMBL28797161

CCCC(CC)NC(=O)Nc1cnc2ccc(-c3cc(C)c(O)c(C)c3)cc2n1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 10/20 0.43
AURKB Q96GD4 6/20 0.43
YES1 P07947 5/20 0.43
HIPK1 Q86Z02 1/20 0.43
PIM1 P11309 2/20 0.42
ABL1 P00519 2/20 0.42
NTRK1 P04629 3/20 0.39
TAS1R3 Q7RTX0 3/20 0.38
TAS1R1 Q7RTX1 3/20 0.38
PIK3CA P42336 8/20 0.38
MAPK8 P45983 3/20 0.37
MAPK9 P45984 3/20 0.37
MAPK10 P53779 3/20 0.37
EGFR P00533 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL629147 0.95 MAPK1 (0.46) MAPK1AURKBYES1HIPK1PIM1
SCHEMBL628841 0.87 MAPK1 (0.45) MAPK1AURKBYES1HIPK1PIM1
SCHEMBL629704 0.84 ABL1 (0.45) MAPK1AURKBYES1HIPK1PIM1
SCHEMBL629121 0.82 MAPK1 (0.51) MAPK1AURKBYES1HIPK1PIM1
SCHEMBL629647 0.82 MAPK1 (0.42) MAPK1AURKBYES1HIPK1PIM1
SCHEMBL630421 0.82 MAPK1 (0.42) MAPK1AURKBYES1HIPK1PIM1
SCHEMBL629037 0.82 MAPK1 (0.61) MAPK1AURKBYES1HIPK1PIM1
SCHEMBL629296 0.81 MAPK1 (0.46) MAPK1AURKBYES1HIPK1PIM1
SCHEMBL629176 0.81 MAPK1 (0.49) MAPK1AURKBYES1HIPK1PIM1
SCHEMBL629375 0.80 MAPK1 (0.48) MAPK1AURKBYES1HIPK1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102378758-A Quinoxaline derivatives and their use for treating benign and malignant tumour disorders AETERNA ZENTARIS GMBH 2012-03-14 CN disclosed