SCHEMBL28798148

SCHEMBL28798148

Cc1nn(-c2ccccc2C#N)c2cccc(-c3cnc4ccccc4c3)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 8/20 0.47
KDM4E B2RXH2 2/20 0.41
PDE10A Q9Y233 1/20 0.38
PARP10 Q53GL7 1/20 0.36
PARP11 Q9NR21 1/20 0.36
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
GABRA1 P14867 2/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRA2 P47869 2/20 0.35
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27873148 0.85 HSP90AA1 (0.47) HSP90AA1KDM4EGABRA1GABRG2GABRB3
SCHEMBL421583 0.84 HSP90AA1 (0.53) HSP90AA1KDM4EALDH1A1NPC1MAPT
SCHEMBL425541 0.84 HSP90AA1 (0.51) HSP90AA1KDM4EPDE10AALDH1A1NPC1
SCHEMBL2182391 0.79 PDGFRB (0.40) HSP90AA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1394528 0.78 HSP90AA1 (0.52) HSP90AA1
SCHEMBL1394538 0.77 HSP90AA1 (0.53) HSP90AA1KDM4EALDH1A1GAAHPGD
SCHEMBL418796 0.77 HSP90AA1 (0.53) HSP90AA1
SCHEMBL421243 0.76 HSP90AA1 (0.62) HSP90AA1
SCHEMBL420425 0.76 HSP90AA1 (0.75) HSP90AA1
SCHEMBL420426 0.76 HSP90AA1 (0.75) HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102439003-A Indazole derivatives inhibiting HSP90, compositions containing said derivatives and uses thereof SANOFI AVENTIS 2012-05-02 CN disclosed