SCHEMBL28798340

SCHEMBL28798340

COc1cc(N2CCOCC2)nc(Nc2ncnc3cc(OC)c(N)cc23)n1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.47
EGFR P00533 6/20 0.47
CYP2C19 P33261 1/20 0.46
KDR P35968 5/20 0.45
KDM4E B2RXH2 1/20 0.44
EPHA2 P29317 3/20 0.44
SRC P12931 4/20 0.43
ERBB2 P04626 1/20 0.43
EPHB4 P54760 1/20 0.42
AURKA O14965 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.41
KCNH2 Q12809 1/20 0.41
MAPK14 Q16539 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29713896 1.00 PDE10A (0.47) PDE10AEGFRCYP2C19KDRKDM4E
SCHEMBL28798349 0.94 PDE10A (0.50) PDE10AEGFRKDRKDM4EEPHA2
SCHEMBL28798338 0.90 EGFR (0.50) PDE10AEGFRKDRKDM4EEPHA2
SCHEMBL29713888 0.90 EGFR (0.50) PDE10AEGFRKDRKDM4EEPHA2
SCHEMBL28798364 0.87 EGFR (0.49) PDE10AEGFRKDRKDM4EEPHA2
SCHEMBL29713885 0.87 EGFR (0.49) PDE10AEGFRKDRKDM4EEPHA2
SCHEMBL29713901 0.85 EGFR (0.49) PDE10AEGFRCYP2C19KDRKDM4E
SCHEMBL28798381 0.85 EGFR (0.49) PDE10AEGFRCYP2C19KDRKDM4E
SCHEMBL28798405 0.83 PDE10A (0.47) PDE10AEGFRKDRKDM4EEPHA2
SCHEMBL30090586 0.82 CYP2C19 (0.46) PDE10AEGFRCYP2C19KDRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114835683-A Quinazoline-4, 6-diamine compound containing morpholinyl aromatic heterocycle and preparation method thereof 江苏食品药品职业技术学院 2022-08-02 CN disclosed