SCHEMBL28800673

SCHEMBL28800673

ON(O)c1ncnc2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.58
PI4KA P42356 1/20 0.50
PI4K2B Q8TCG2 1/20 0.50
PI4K2A Q9BTU6 1/20 0.50
PI4KB Q9UBF8 1/20 0.50
PDE4A P27815 1/20 0.50
PDE4B Q07343 1/20 0.50
PDE4C Q08493 1/20 0.50
PDE4D Q08499 1/20 0.50
ADORA2A P29274 2/20 0.47
ALDH1A1 P00352 1/20 0.43
HTT P42858 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ABCG2 Q9UNQ0 2/20 0.43
DAPK3 O43293 1/20 0.43
MAP4K4 O95819 1/20 0.43
ABL1 P00519 1/20 0.43
ERBB2 P04626 1/20 0.43
PIM1 P11309 1/20 0.43
PRKACA P17612 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4030057 0.81 EGFR (0.65) EGFRPI4KAPI4K2BPI4K2API4KB
SCHEMBL2184445 0.79 EGFR (0.68) EGFRPI4KAPI4K2BPI4K2API4KB
Hydrochloric Acid SCHEMBL14775621 0.78 EGFR (0.66) EGFRPI4KAPI4K2BPI4K2API4KB
SCHEMBL8900055 0.76 EGFR (0.69) EGFRPI4KAPI4K2BPI4K2API4KB
SCHEMBL11013925 0.75 HTT (0.61) EGFRPI4KAPI4K2BPI4K2API4KB
Hydrochloric Acid SCHEMBL6039704 0.75 EGFR (0.67) EGFRPI4KAPI4K2BPI4K2API4KB
SCHEMBL4424934 0.73 EGFR (0.47) EGFRPI4KAPI4K2BPI4K2API4KB
SCHEMBL21415554 0.73 EGFR (0.60) EGFRPI4KAPI4K2BPI4K2API4KB
Hydrochloric Acid SCHEMBL8375173 0.73 HTT (0.59) EGFRPI4KAPI4K2BPI4K2API4KB
SCHEMBL3109912 0.73 EGFR (1.00) EGFRHDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102827087-B Synthetic method of erlotinib CHENGDU INST BIOLOGY CAS 2015-03-25 CN disclosed
CN-102827087-A Synthetic method of erlotinib CHENGDU INST BIOLOGY CAS 2012-12-19 CN disclosed