Benzene

Benzene

SCHEMBL28800797

Nc1ccc2nc(N)ncc2c1.c1ccccc1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.53
LCK P06239 2/20 0.53
KDR P35968 2/20 0.53
JAK3 P52333 1/20 0.53
MAPK14 Q16539 1/20 0.53
ALDH1A1 P00352 3/20 0.50
HSD17B10 Q99714 3/20 0.50
KDM4E B2RXH2 2/20 0.50
ATM Q13315 2/20 0.50
CASP1 P29466 2/20 0.50
HTT P42858 2/20 0.50
TP53 P04637 1/20 0.50
HSP90AA1 P07900 1/20 0.50
HSP90AB1 P08238 1/20 0.50
MAPT P10636 1/20 0.50
TSHR P16473 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
PLAU P00749 1/20 0.48
CSNK1D P48730 1/20 0.47
CSNK1E P49674 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30912753 0.96 EGFR (0.57) EGFRLCKKDRJAK3MAPK14
SCHEMBL610225 0.96 EGFR (0.57) EGFRLCKKDRJAK3MAPK14
Benzene SCHEMBL27889171 0.81 LCK (0.50) LCKKDRJAK3MAPK14ALDH1A1
SCHEMBL5494272 0.81 LCK (0.58) EGFRLCKKDRJAK3MAPK14
SCHEMBL5488838 0.80 MAP4K4 (0.61) LCKKDRJAK3MAPK14ALDH1A1
SCHEMBL2741576 0.79 LCK (0.65) LCKKDRJAK3MAPK14KIT
SCHEMBL24150165 0.79 HTT (0.58) EGFRLCKKDRJAK3MAPK14
SCHEMBL3191937 0.78 TLR9 (0.57) EGFRALDH1A1HSD17B10KDM4EATM
SCHEMBL2130969 0.76 PIK3CG (0.53) LCKKDRJAK3MAPK14KDM4E
SCHEMBL2632884 0.76 LCK (0.57) LCKKDRJAK3MAPK14ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102850397-B Multi-target antitumor compounds and preparation method and application thereof UNIV BEIJING 2015-02-18 CN claimed
CN-102850397-A Multi-target antitumor compounds and preparation method and application thereof UNIV BEIJING 2013-01-02 CN claimed
CN-102850397-B Multi-target antitumor compounds and preparation method and application thereof UNIV BEIJING 2015-02-18 CN disclosed
CN-102850397-A Multi-target antitumor compounds and preparation method and application thereof UNIV BEIJING 2013-01-02 CN disclosed