SCHEMBL28801137

SCHEMBL28801137

Cc1cc(Br)cn2ncc(C(=O)ON)c12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.34
PLAU P00749 1/20 0.33
ELANE P08246 1/20 0.33
KMT2A Q03164 3/20 0.33
TSHR P16473 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 3/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
EGFR P00533 1/20 0.31
ERBB2 P04626 1/20 0.31
KDR P35968 1/20 0.31
EPHB3 P54753 1/20 0.30
MAPK14 Q16539 2/20 0.30
PKM P14618 2/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
TYK2 P29597 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24329437 0.87 KMT2A (0.43) KMT2ATSHRMEN1ALDH1A1HPGD
SCHEMBL29066241 0.82 RXFP1 (0.43) RXFP1PLAUELANEALDH1A1EPHB3
SCHEMBL16914025 0.75 KMT2A (0.42) KMT2ATSHRMEN1ALDH1A1HPGD
SCHEMBL28801147 0.74 EPHB3 (0.53) ALDH1A1HPGDRAB9AEPHB3SMN1; SMN2
SCHEMBL20909486 0.74 TSHR (0.45) KMT2ATSHRMEN1ALDH1A1HPGD
SCHEMBL23501291 0.73 TSHR (0.44) KMT2ATSHRMEN1ALDH1A1HPGD
SCHEMBL1907994 0.72 KMT2A (0.42) KMT2AMEN1KDRMAPK14PKM
SCHEMBL31393197 0.72 TSHR (0.43) KMT2ATSHRMEN1ALDH1A1HPGD
SCHEMBL25287018 0.71 EGFR (0.43) KMT2ATSHRMEN1ALDH1A1HPGD
SCHEMBL23501300 0.69 SIK1 (0.38) TSHRALDH1A1HPGDEGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884050-B Tetrahydroisoquinoline derivatives UCB生物制药私人有限公司 2022-07-05 CN disclosed