SCHEMBL28801576

SCHEMBL28801576

COc1c(C(C)C)cnn1-c1c(Cl)cccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.38
NPBWR1 P48145 9/20 0.37
MCHR1 Q99705 8/20 0.37
GAA P10253 1/20 0.36
MAPK14 Q16539 3/20 0.34
ALDH1A1 P00352 2/20 0.33
KMT2A Q03164 2/20 0.33
NPC1 O15118 1/20 0.33
S1PR4 O95977 1/20 0.33
MAPT P10636 1/20 0.33
S1PR1 P21453 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
PAX8 Q06710 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
P2RX7 Q99572 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1097175 0.76 NR1H4 (0.41) NR1H4NPBWR1MCHR1GAAMAPK14
SCHEMBL2774647 0.76 NR1H4 (0.45) NR1H4NPBWR1MCHR1MAPK14ALDH1A1
SCHEMBL1096331 0.75 NR1H4 (0.44) NR1H4NPBWR1MCHR1MAPK14ALDH1A1
SCHEMBL1095989 0.75 NR1H4 (0.46) NR1H4NPBWR1MCHR1MAPK14KMT2A
SCHEMBL20094462 0.75 NR1H4 (0.40) NR1H4NPBWR1MCHR1MAPK14ALDH1A1
SCHEMBL27896015 0.73 NR1H4 (0.39) NR1H4NPBWR1MCHR1SMN1; SMN2P2RX7
SCHEMBL27896299 0.72 NR1H4 (0.43) NR1H4MAPK14ALDH1A1
SCHEMBL21340190 0.72 NR1H4 (0.43) NR1H4MAPK14
SCHEMBL26272107 0.72 NR1H4 (0.43) NR1H4NPBWR1MCHR1MAPK14P2RX7
SCHEMBL21849905 0.68 PRMT5 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101743232-B Compounds and methods for modulating fxr LILLY CO ELI 2013-03-06 CN disclosed