SCHEMBL28802401

SCHEMBL28802401

CC(c1nc2ccccc2cc1CN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Cc1nnn[nH]1)N(C)C1CCCC1

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 9/20 0.32
TACR2 P21452 2/20 0.32
BACE1 P56817 1/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
TSHR P16473 2/20 0.31
NPSR1 Q6W5P4 2/20 0.31
HSD17B10 Q99714 2/20 0.31
USP2 O75604 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27902067 0.87 TACR1 (0.33) TACR1TACR2BACE1
SCHEMBL27901998 0.86 TACR1 (0.42) TACR1TACR2BACE1
SCHEMBL5624144 0.83
SCHEMBL27901982 0.82 TACR1 (0.43) TACR1BACE1
SCHEMBL5624134 0.79 BCHE (0.32) TACR1TACR2
SCHEMBL5626484 0.77 TACR1 (0.40) TACR1BACE1
SCHEMBL27919744 0.77 TACR1 (0.32) TACR1TACR2BACE1
SCHEMBL27919745 0.77 CETP (0.39) TACR1
SCHEMBL27902000 0.76 TACR1 (0.32) TACR1TACR2BACE1
SCHEMBL27902051 0.76 BACE1 (0.32) TACR1TACR2BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103102303-A Benzylamine derivatives as CETP inhibitors REDDY US THERAPEUTICS INC 2013-05-15 CN disclosed