SCHEMBL28802455

SCHEMBL28802455

CN(C(=O)c1cc(C(N)=O)cc(CCl)n1)C1CC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.38
SMYD3 Q9H7B4 3/20 0.36
SYK P43405 2/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
POLB P06746 1/20 0.34
S1PR1 P21453 1/20 0.34
DPP4 P27487 2/20 0.33
DPP9 Q86TI2 2/20 0.33
DPP7 Q9UHL4 2/20 0.33
F2 P00734 2/20 0.33
DPP8 Q6V1X1 1/20 0.33
ALOX5 P09917 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19641703 0.88 BRD4 (0.39) BRD4SMYD3SYKNPC1RAB9A
SCHEMBL28802499 0.82 BRD4 (0.62) BRD4NPC1RAB9A
SCHEMBL19641880 0.81 BRD4 (0.49) BRD4NPC1RAB9A
SCHEMBL28802495 0.80 SYK (0.36) SMYD3SYKNPC1RAB9APOLB
SCHEMBL28802480 0.80 BRD4 (0.62) BRD4NPC1RAB9A
SCHEMBL19642320 0.79 BRD4 (0.45) BRD4SMYD3NPC1RAB9A
SCHEMBL29831147 0.79 BRD4 (0.45) BRD4SMYD3NPC1RAB9A
SCHEMBL28802468 0.79 BRD4 (0.61) BRD4NPC1RAB9A
SCHEMBL19641713 0.79 BRD4 (0.47) BRD4NPC1RAB9ADPP4DPP9
SCHEMBL19641665 0.79 BRD4 (0.49) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109153646-B Pyridine dicarboxamide derivatives as bromodomain inhibitors 葛兰素史克知识产权第二有限公司 2022-08-02 CN disclosed