SCHEMBL28806325

SCHEMBL28806325

CC(C)(C)C(=O)ON1CCC(n2cc(NC(=O)c3ccc(-n4cc(-c5n[nH]c6ccccc56)nn4)cc3)cn2)CC1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 6/20 0.41
DYRK1A Q13627 6/20 0.41
CLK2 P49760 1/20 0.41
CLK3 P49761 1/20 0.41
FGFR1 P11362 3/20 0.39
DDR2 Q16832 3/20 0.39
ROCK1 Q13464 7/20 0.39
ITK Q08881 1/20 0.37
ROCK2 O75116 1/20 0.37
NAMPT P43490 1/20 0.36
RPS6KA2 Q15349 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27926193 0.97 GSK3B (0.39) GSK3BDYRK1ACLK2CLK3FGFR1
SCHEMBL9952339 0.90 DDB1 (0.44) GSK3BDYRK1ACLK2CLK3FGFR1
SCHEMBL9952422 0.89 GSK3B (0.51) GSK3BDYRK1ACLK2CLK3FGFR1
SCHEMBL9952674 0.87 DDB1 (0.42) GSK3BDYRK1ACLK2CLK3FGFR1
SCHEMBL10194961 0.86 GSK3B (0.46) GSK3BDYRK1ACLK2CLK3FGFR1
SCHEMBL10195389 0.86 GSK3B (0.49) GSK3BDYRK1ACLK2CLK3FGFR1
Tert-Butyl Formate SCHEMBL28806326 0.85 GSK3B (0.45) GSK3BDYRK1ACLK2CLK3FGFR1
Hydrochloric Acid SCHEMBL15312398 0.85 GSK3B (0.48) GSK3BDYRK1ACLK2CLK3FGFR1
SCHEMBL15312572 0.84 GSK3B (0.40) GSK3BDYRK1ACLK2CLK3FGFR1
SCHEMBL10195391 0.83 GSK3B (0.46) GSK3BDYRK1ACLK2CLK3FGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103429585-A Indazolyl triazole derivatives as interleukin-1 receptor associated kinase inhibitors MERCK SERONO SA 2013-12-04 CN disclosed