SCHEMBL28809248

SCHEMBL28809248

O=C(Nc1ccncc1)c1c[nH]c2ccc(-c3cccnc3F)cc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKE Q14164 1/20 0.50
TBK1 Q9UHD2 1/20 0.50
DYRK1A Q13627 3/20 0.49
CLK2 P49760 1/20 0.49
CLK3 P49761 1/20 0.49
ROCK1 Q13464 3/20 0.45
HTR2C P28335 3/20 0.44
KMT2A Q03164 1/20 0.44
PRKCI P41743 1/20 0.44
ALDH1A1 P00352 1/20 0.44
NR4A2 P43354 1/20 0.43
ROCK2 O75116 1/20 0.43
MAPT P10636 1/20 0.43
BACE1 P56817 1/20 0.43
NHERF1 O14745 2/20 0.43
HTT P42858 1/20 0.43
WNT1 P04628 1/20 0.42
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29753935 1.00 IKBKE (0.50) IKBKETBK1DYRK1ACLK2CLK3
SCHEMBL29753996 0.85 DYRK1A (0.48) DYRK1ACLK2CLK3ROCK1ROCK2
SCHEMBL28810265 0.85 DYRK1A (0.48) DYRK1ACLK2CLK3ROCK1ROCK2
SCHEMBL29754130 0.83 DHODH (0.54) DYRK1ANR4A2MAPT
SCHEMBL28947575 0.83 DHODH (0.54) DYRK1ANR4A2MAPT
SCHEMBL23533877 0.81 DYRK1A (0.70) DYRK1ACLK2CLK3WNT1
SCHEMBL29753923 0.81 DYRK1A (0.70) DYRK1ACLK2CLK3WNT1
SCHEMBL28811003 0.79 DYRK1A (0.51) DYRK1ACLK2CLK3KMT2AALDH1A1
SCHEMBL29754069 0.79 BACE1 (0.60) DYRK1AKMT2AALDH1A1MAPTBACE1
SCHEMBL28811002 0.79 DYRK1A (0.51) DYRK1ACLK2CLK3KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114867718-A Novel indazole derivative and use thereof 韩国化学研究院 2022-08-05 CN disclosed