SCHEMBL28816280

SCHEMBL28816280

CCOC(=O)c1nc(-c2ccc(F)cc2)no1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.68
KMT2A Q03164 4/20 0.49
POLB P06746 1/20 0.49
TRPM8 Q7Z2W7 1/20 0.49
NPC1 O15118 3/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
GABRA2 P47869 1/20 0.48
GABRB2 P47870 1/20 0.48
TPH1 P17752 2/20 0.46
GRM6 O15303 1/20 0.46
MAPT P10636 5/20 0.46
MEN1 O00255 3/20 0.46
ALDH1A1 P00352 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
SLC26A6 Q9BXS9 1/20 0.45
MAPK1 P28482 2/20 0.45
KDM4E B2RXH2 1/20 0.45
PKM P14618 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3233714 0.89 HTT (0.71) HTTKMT2ATRPM8NPC1RAB9A
SCHEMBL3230760 0.86 HTT (0.68) HTTKMT2ATRPM8NPC1RAB9A
SCHEMBL3335119 0.86 HTT (0.72) HTTPOLBNPC1RAB9ASMN1; SMN2
SCHEMBL8593668 0.86 HTT (0.68) HTTKMT2APOLBNPC1SMN1; SMN2
SCHEMBL28816317 0.86 HTT (0.68) HTTKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL2554648 0.86 HTT (0.67) HTTKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL28816242 0.85 KMT2A (0.53) HTTKMT2APOLBNPC1RAB9A
SCHEMBL28816269 0.85 HTT (0.64) HTTKMT2ASMN1; SMN2MAPTMEN1
SCHEMBL4528391 0.84 HTT (0.66) HTTKMT2APOLBNPC1RAB9A
SCHEMBL22619755 0.84 HTT (0.66) HTTTRPM8NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114933573-A 3-substituted-1, 2, 4-oxadiazole-5-carboxylic acid derivative, and preparation method and application thereof 贵州大学 2022-08-23 CN claimed
CN-114933573-B 3-substituted-1, 2, 4-oxadiazole-5-carboxylic acid derivative, and preparation method and application thereof 贵州大学 2023-10-20 CN disclosed
CN-114933573-A 3-substituted-1, 2, 4-oxadiazole-5-carboxylic acid derivative, and preparation method and application thereof 贵州大学 2022-08-23 CN disclosed