SCHEMBL28819985

SCHEMBL28819985

N#Cc1cnc2[nH]cc(Cc3cccnc3NCc3cnccc3C(F)(F)F)c2c1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.53
CYP2C19 P33261 1/20 0.52
CDC7 O00311 1/20 0.41
MAP4K4 O95819 1/20 0.41
PIM1 P11309 1/20 0.41
PRKACA P17612 1/20 0.41
CDK2 P24941 1/20 0.41
GSK3B P49841 1/20 0.41
HIPK2 Q9H2X6 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.41
PRKCQ Q04759 9/20 0.40
PRKCD Q05655 6/20 0.40
GPR84 Q9NQS5 1/20 0.39
CSF1R P07333 1/20 0.39
KIT P10721 1/20 0.39
CYP2C9 P11712 3/20 0.38
PTK2 Q05397 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1887646 0.83 CYP3A4 (0.77) CYP3A4CYP2C19CSF1RKITCYP2C9
SCHEMBL28018895 0.82 CYP2C9 (0.55) CYP3A4CYP2C19PRKCQCSF1RKIT
SCHEMBL28018897 0.80 CYP3A4 (0.58) CYP3A4CYP2C19GPR84CSF1RKIT
SCHEMBL28108746 0.79 CYP3A4 (0.54) CYP3A4CYP2C19GPR84CSF1RKIT
SCHEMBL28108734 0.78 CYP3A4 (0.56) CYP3A4CYP2C19CSF1RKITCYP2C9
SCHEMBL28018398 0.75 CYP2C9 (0.55) CYP3A4CYP2C19CSF1RCYP2C9
SCHEMBL1267406 0.75 CYP3A4 (0.60) CYP3A4CYP2C19CDC7MAP4K4PIM1
SCHEMBL1890594 0.73 CYP3A4 (0.60) CYP3A4CYP2C19CDC7MAP4K4PIM1
SCHEMBL1883948 0.72 CYP3A4 (0.77) CYP3A4CYP2C19CDC7MAP4K4PIM1
SCHEMBL1881856 0.71 CYP3A4 (0.66) CYP3A4CYP2C19CSF1RKITCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104703623-A Compounds and methods for kinase modulation, and indications therefor PLEXXIKON INC 2015-06-10 CN disclosed