SCHEMBL28820139

SCHEMBL28820139

COc1cc2ncnc([NH+]([O-])c3ccc(F)c(Cl)c3)c2cc1OCCCN1CCOCC1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.68
KDR P35968 5/20 0.68
FLT4 P35916 3/20 0.68
KIT P10721 3/20 0.68
BRAF P15056 2/20 0.68
ERBB2 P04626 2/20 0.68
SRC P12931 2/20 0.68
RET P07949 2/20 0.68
CIT O14578 1/20 0.68
GAK O14976 1/20 0.68
EPHB6 O15197 1/20 0.68
ABCC4 O15439 1/20 0.68
DAPK3 O43293 1/20 0.68
RIPK2 O43353 1/20 0.68
NR1I2 O75469 1/20 0.68
RPS6KA4 O75676 1/20 0.68
STK17B O94768 1/20 0.68
STK10 O94804 1/20 0.68
PRKD3 O94806 1/20 0.68
ABCB11 O95342 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22594686 0.83 KDR (0.70) EGFRKDRFLT4KITBRAF
SCHEMBL13319080 0.82 EGFR (0.71) EGFRKDRFLT4KITBRAF
Gefitinib SCHEMBL7866 0.81 EGFR (1.00) EGFRKDRFLT4KITBRAF
Gefitinib SCHEMBL29351046 0.81 EGFR (1.00) EGFRKDRFLT4KITBRAF
Gefitinib SCHEMBL29351336 0.81 EGFR (1.00) EGFRKDRFLT4KITBRAF
SCHEMBL1734701 0.81 EGFR (1.00) EGFRKDRFLT4KITBRAF
Gefitinib SCHEMBL465143 0.81 EGFR (1.00) EGFRKDRFLT4KITBRAF
SCHEMBL23258972 0.80 EGFR (0.80) EGFRKDRFLT4KITBRAF
Gefitinib SCHEMBL2770155 0.80 EGFR (0.98) EGFRKDRFLT4KITBRAF
Gefitinib SCHEMBL30887946 0.80 EGFR (0.98) EGFRKDRFLT4KITBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104817506-A Quinazoline nitrogen oxide SHANGDONG NEW TIME PHARM PROD 2015-08-05 CN disclosed