SCHEMBL28821900

SCHEMBL28821900

NC(=O)c1ccc2oc(N3CCCC3)nc2c1

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.49
FAAH O00519 1/20 0.48
CNR2 P34972 2/20 0.47
HRH3 Q9Y5N1 1/20 0.47
PTGES O14684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28821901 0.99 HRH3 (0.48) HDAC6FAAHCNR2HRH3PTGES
SCHEMBL22227676 0.89 CNR2 (0.50) HDAC6FAAHCNR2
SCHEMBL20296248 0.88 KDM4E (0.51) HDAC6
SCHEMBL18344206 0.87 NPC1 (0.55) HDAC6FAAHCNR2PTGES
SCHEMBL20296406 0.87 HDAC6 (0.53) HDAC6HRH3PTGES
SCHEMBL20296288 0.87 CNR2 (0.52) HDAC6CNR2
SCHEMBL18344187 0.86 NPC1 (0.57) HDAC6FAAHCNR2PTGES
SCHEMBL20296478 0.86 HDAC6 (0.45) HDAC6
SCHEMBL20296414 0.85 HDAC6 (0.45) HDAC6CNR2HRH3PTGES
SCHEMBL3468711 0.85 HRH3 (0.52) HDAC6CNR2HRH3PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107743483-B NADPH oxidase 4 inhibitors 埃科特莱茵药品有限公司 2022-01-28 CN claimed
CN-107743483-B NADPH oxidase 4 inhibitors 埃科特莱茵药品有限公司 2022-01-28 CN disclosed