SCHEMBL28822962

SCHEMBL28822962

Cc1ccc(-c2nc(N)c(C#N)nc2-c2ccc(C)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.53
ADORA1 P30542 4/20 0.51
ADORA2A P29274 4/20 0.51
USP8 P40818 2/20 0.47
NPSR1 Q6W5P4 4/20 0.45
MYC P01106 1/20 0.45
WDR5 P61964 1/20 0.45
KDM4E B2RXH2 4/20 0.42
MAPT P10636 3/20 0.42
LMNA P02545 2/20 0.42
MAPK1 P28482 2/20 0.42
XBP1 P17861 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ADORA2B P29275 1/20 0.42
TDP1 Q9NUW8 2/20 0.42
KMT2A Q03164 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
USP7 Q93009 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28949046 0.92 KDM4E (0.47) ERBB2ADORA1ADORA2AUSP8NPSR1
SCHEMBL28823032 0.89 ADORA1 (0.55) ERBB2ADORA1ADORA2ANPSR1MYC
SCHEMBL2681245 0.87 ERBB2 (0.61) ERBB2ADORA1ADORA2AUSP8NPSR1
SCHEMBL14545408 0.82 ERBB2 (0.53) ERBB2ADORA1ADORA2AUSP8MYC
SCHEMBL28823015 0.81 USP8 (0.58) ERBB2ADORA1ADORA2AUSP8KDM4E
SCHEMBL28822957 0.81 ADORA1 (0.56) ADORA1ADORA2AUSP8KDM4EADORA2B
SCHEMBL28822967 0.81 ADORA1 (0.56) ADORA1ADORA2AUSP8KDM4EADORA2B
SCHEMBL21722354 0.79 ADORA2A (0.58) ERBB2ADORA1ADORA2AKDM4EMAPT
SCHEMBL4684019 0.79 ERBB2 (0.53) ERBB2ADORA1ADORA2AUSP8NPSR1
SCHEMBL15106376 0.78 KDM4E (0.39) ERBB2ADORA1ADORA2ANPSR1MYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114644597-B Tetra-substituted pyrazine derivative and preparation method and application thereof 南京农业大学 2023-11-21 CN claimed
CN-114644597-A Tetra-substituted pyrazine derivative and preparation method and application thereof 南京农业大学 2022-06-21 CN claimed
CN-114644597-B Tetra-substituted pyrazine derivative and preparation method and application thereof 南京农业大学 2023-11-21 CN disclosed
CN-114644597-A Tetra-substituted pyrazine derivative and preparation method and application thereof 南京农业大学 2022-06-21 CN disclosed