SCHEMBL28833581

SCHEMBL28833581

[CH2][C@@H](Cc1ccccc1)C(=O)NCC(=O)OCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
ABCC3 O15438 1/20 0.60
NR1I2 O75469 1/20 0.60
ABCB11 O95342 1/20 0.60
NR3C1 P04150 1/20 0.60
RARG P13631 1/20 0.60
CNR1 P21554 1/20 0.60
OPRK1 P41145 1/20 0.60
NR1H2 P55055 1/20 0.60
PPARA Q07869 1/20 0.60
NR1H3 Q13133 1/20 0.60
NR1I3 Q14994 1/20 0.60
L3MBTL1 Q9Y468 2/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPK1 P28482 1/20 0.49
MEN1 O00255 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22539312 0.83 CYP1A2 (0.64) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL19844611 0.83 CYP3A4 (0.64) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7105553 0.82 CYP1A2 (0.70) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7107731 0.82 CYP1A2 (0.70) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL28095683 0.82 MME (0.62) ALDH1A1MAPK1MEN1KMT2AHPGD
SCHEMBL28095685 0.82 MME (0.62) ALDH1A1MAPK1MEN1KMT2AHPGD
SCHEMBL19844612 0.81 CYP2D6 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7107227 0.81 CYP1A2 (0.68) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7694738 0.81 CYP1A2 (0.68) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL10694679 0.81 CYP1A2 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103739531-B Novel aminoacid derivate, its preparation method and therapeutic use 领先药物公司 2016-09-14 CN disclosed