SCHEMBL28833844

SCHEMBL28833844

NC(=O)OC1CCN(c2ncnc3c(F)c(-c4ccccc4F)c(Cl)cc23)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KRAS P01116 8/20 0.54
EGFR P00533 1/20 0.54
HMOX2 P30519 1/20 0.54
CRYZ Q08257 1/20 0.54
VAT1 Q99536 1/20 0.54
RTN4 Q9NQC3 1/20 0.54
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
KIT P10721 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CNR1 P21554 6/20 0.37
CNR2 P34972 4/20 0.37
PDE10A Q9Y233 1/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29888384 0.85 KRAS (0.49) KRASEGFRHMOX2CRYZVAT1
SCHEMBL23415237 0.85 KRAS (0.49) KRASEGFRHMOX2CRYZVAT1
Hydrochloric Acid SCHEMBL29888512 0.84 KRAS (0.49) KRASEGFRHMOX2CRYZVAT1
Hydrochloric Acid SCHEMBL23415303 0.84 KRAS (0.49) KRASEGFRHMOX2CRYZVAT1
SCHEMBL23415476 0.84 KRAS (0.51) KRASEGFRHMOX2CRYZVAT1
SCHEMBL29901300 0.84 KRAS (0.51) KRASEGFRHMOX2CRYZVAT1
SCHEMBL23415473 0.83 KRAS (0.50) KRASEGFRHMOX2CRYZVAT1
SCHEMBL29888636 0.83 KRAS (0.50) KRASEGFRHMOX2CRYZVAT1
SCHEMBL23415339 0.83 KRAS (0.51) KRASEGFRHMOX2CRYZVAT1
SCHEMBL16646882 0.81 KRAS (0.77) KRASEGFRHMOX2CRYZVAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114980976-A Covalent RAS inhibitors and uses thereof 锐新医药公司 2022-08-30 CN disclosed