SCHEMBL28834249

SCHEMBL28834249

COc1cc2nccc(OC3CCN(C(=O)OC(C)(C)C)C3)c2cc1OC

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 4/20 0.60
PIK3CA P42336 3/20 0.60
PIK3CB P42338 3/20 0.60
PIK3CG P48736 3/20 0.60
PDE4B Q07343 3/20 0.52
PDE4A P27815 2/20 0.52
PDE4C Q08493 2/20 0.52
PDE4D Q08499 2/20 0.52
BRAF P15056 1/20 0.51
KRAS P01116 3/20 0.49
SOS1 Q07889 3/20 0.49
IDO1 P14902 1/20 0.49
EGFR P00533 4/20 0.47
ERBB2 P04626 1/20 0.47
NSD2 O96028 1/20 0.47
PDE10A Q9Y233 3/20 0.46
PDE3B Q13370 2/20 0.45
PDE3A Q14432 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29933502 1.00 PIK3CD (0.60) PIK3CDPIK3CAPIK3CBPIK3CGPDE4B
SCHEMBL28834247 1.00 PIK3CD (0.60) PIK3CDPIK3CAPIK3CBPIK3CGPDE4B
SCHEMBL25130494 0.91 PIK3CD (0.56) PIK3CDPIK3CAPIK3CBPIK3CGPDE4B
SCHEMBL28834207 0.88 PIK3CD (0.58) PIK3CDPIK3CAPIK3CBPIK3CGPDE4B
SCHEMBL29933652 0.88 PIK3CD (0.58) PIK3CDPIK3CAPIK3CBPIK3CGPDE4B
SCHEMBL28834206 0.88 PIK3CD (0.58) PIK3CDPIK3CAPIK3CBPIK3CGPDE4B
SCHEMBL23360649 0.86 PIK3CD (0.55) PIK3CDPIK3CAPIK3CBPIK3CGKRAS
SCHEMBL23360651 0.86 PIK3CD (0.55) PIK3CDPIK3CAPIK3CBPIK3CGKRAS
SCHEMBL25130570 0.84 PDE4B (0.55) PIK3CDPIK3CAPIK3CBPIK3CGPDE4B
SCHEMBL18497822 0.84 IRAK4 (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114867719-B Pyrrolidine and piperidine compounds 柳韩洋行 2024-06-25 CN disclosed
CN-114867719-A Pyrrolidine and piperidine compounds 柳韩洋行 2022-08-05 CN disclosed