SCHEMBL28835246

SCHEMBL28835246

NC(=O)c1cc(N2CCC(NC(=O)O)C2)cnc1Oc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BTK Q06187 13/20 0.55
CA12 O43570 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA4 P22748 2/20 0.46
CA7 P43166 2/20 0.46
CA9 Q16790 2/20 0.46
SYK P43405 1/20 0.43
RPS6KB1 P23443 1/20 0.41
USP30 Q70CQ3 2/20 0.40
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16670822 0.94 BTK (0.56) BTKCA12CA1CA2CA4
SCHEMBL16670054 0.90 BTK (0.70) BTK
SCHEMBL16670664 0.89 BTK (0.56) BTKCA12CA1CA2CA4
SCHEMBL16676753 0.89 BTK (0.52) BTKCA12CA1CA2CA4
SCHEMBL18044925 0.89 BTK (0.56) BTKCA12CA1CA2CA4
SCHEMBL16670904 0.87 BTK (0.49) BTKCA12CA1CA2CA4
SCHEMBL16670710 0.86 BTK (0.45) BTKSYK
SCHEMBL16671599 0.85 BTK (0.71) BTK
SCHEMBL16671450 0.84 BTK (0.64) BTKSYK
SCHEMBL16671485 0.84 BTK (0.44) BTKSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105939998-B Heteroaryl compound and application thereof as BTK inhibitor 默克专利有限公司 2019-04-16 CN disclosed
CN-105939998-A Heteroaryl compounds as btk inhibitors and uses thereof 默克专利有限公司 2016-09-14 CN disclosed