SCHEMBL28840394

SCHEMBL28840394

COC(=O)c1cncc(OCC(F)F)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.51
GRM5 P41594 1/20 0.48
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
SIRT2 Q8IXJ6 2/20 0.42
SIRT3 Q9NTG7 2/20 0.42
SIRT1 Q96EB6 1/20 0.42
CYP2A6 P11509 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KDM4E B2RXH2 1/20 0.40
PRMT5 O14744 1/20 0.39
WDR77 Q9BQA1 1/20 0.39
P2RX3 P56373 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
S1PR1 P21453 1/20 0.37
MAPK1 P28482 1/20 0.37
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16319115 0.87 ATM (0.53) ATMGRM5CYP11B1CYP11B2SIRT2
SCHEMBL23167202 0.83 ATM (0.56) ATMGRM5CYP11B1CYP11B2SIRT2
SCHEMBL30281264 0.83 HCAR2 (0.47) SIRT2ALDH1A1KDM4EP2RX3CYP2C9
SCHEMBL14004766 0.83 ATM (0.49) ATMGRM5CYP11B1CYP11B2SIRT2
SCHEMBL30281289 0.82 SIRT2 (0.47) SIRT2SIRT3SIRT1
SCHEMBL17781534 0.80 ATM (0.56) ATMGRM5CYP11B1CYP11B2SIRT2
SCHEMBL1806939 0.79 ATM (0.51) ATMGRM5CYP11B1CYP11B2SIRT2
SCHEMBL28060971 0.79 ATM (0.54) ATMGRM5CYP11B1CYP11B2SIRT2
SCHEMBL12524683 0.78 ATM (0.53) ATMGRM5CYP11B1CYP11B2MAPT
SCHEMBL31287098 0.78 ATM (0.53) ATMGRM5CYP11B1CYP11B2SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106478497-A Aryl amine derivatives as TTX S blocker 拉夸里亚创药株式会社 2017-03-08 CN disclosed