SCHEMBL28840580

SCHEMBL28840580

NC(=O)c1cccc2[nH]c(-c3ccc(C(=O)N4CCN(C(=O)c5ccccc5)CC4)cc3)nc12

nearest known ligand 0.84

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.84
DHODH Q02127 4/20 0.84
CHEK2 O96017 1/20 0.64
PARP2 Q9UGN5 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29790489 1.00 PARP1 (0.84) PARP1DHODHCHEK2PARP2
SCHEMBL28840989 0.92 PARP1 (0.82) PARP1DHODHCHEK2PARP2
SCHEMBL28840577 0.91 PARP1 (0.80) PARP1DHODHPARP2
SCHEMBL29790473 0.91 PARP1 (0.80) PARP1DHODHPARP2
SCHEMBL31413270 0.90 PARP1 (0.82) PARP1DHODHPARP2
SCHEMBL28840597 0.90 PARP1 (0.74) PARP1DHODHCHEK2PARP2
SCHEMBL29790486 0.90 PARP1 (0.74) PARP1DHODHCHEK2PARP2
Hydrochloric Acid SCHEMBL31413181 0.89 PARP1 (0.80) PARP1DHODHPARP2
SCHEMBL29790574 0.89 PARP1 (0.76) PARP1DHODHPARP2
SCHEMBL28840603 0.89 PARP1 (0.76) PARP1DHODHPARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114907269-A Benzimidazole-4-carboxamide derivative with piperazine as connecting group 南华大学 2022-08-16 CN disclosed