SCHEMBL28840764

SCHEMBL28840764

O=C(O)Cc1ccc2c(c1)COCC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 3/20 0.46
CA2 P00918 2/20 0.44
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
RXRG P48443 1/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPT P10636 3/20 0.43
HPGD P15428 3/20 0.43
HSD17B10 Q99714 3/20 0.43
GAA P10253 2/20 0.43
RGS12 O14924 1/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
APEX1 P27695 1/20 0.43
THPO P40225 1/20 0.43
BLM P54132 1/20 0.43
GNAI1 P63096 1/20 0.43
PMP22 Q01453 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5173443 0.86 GAA (0.48) AKR1B1CA2RXRARXRBRXRG
SCHEMBL31478167 0.81 AKR1B1 (0.58) AKR1B1CA2RXRARXRBRXRG
SCHEMBL21382554 0.80 PRMT5 (0.40) CA2PRMT5WDR77FFAR4
SCHEMBL3838996 0.79 RXRB (0.62) AKR1B1RXRARXRBRXRGKDM4E
SCHEMBL5527444 0.78 RXRB (0.65) AKR1B1RXRARXRBRXRGKDM4E
SCHEMBL19996854 0.78 RXRB (0.60) AKR1B1RXRARXRBRXRGKDM4E
SCHEMBL9123053 0.76 PRMT5 (0.38) KDM4EHSD17B10PRMT5WDR77
SCHEMBL21382504 0.76 PRMT5 (0.38) PRMT5WDR77
SCHEMBL28840799 0.76 PRMT5 (0.38) PRMT5WDR77
SCHEMBL26574191 0.76 KDM4E (0.45) CA2KDM4EMAPTHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114907389-A Boronic acid derivatives 首药控股(北京)股份有限公司 2022-08-16 CN disclosed