SCHEMBL28843641

SCHEMBL28843641

Fc1cccc(F)c1.N#Cc1ccccc1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.41
PGR P06401 2/20 0.41
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
ESR2 Q92731 2/20 0.39
TSHR P16473 2/20 0.38
LMNA P02545 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
ALOX12 P18054 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
CA12 O43570 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
NQO2 P16083 1/20 0.37
PTGS1 P23219 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28161686 0.84 ESR1 (0.43) ARPGRESR2LMNAMEN1
SCHEMBL29392995 0.83
SCHEMBL27875336 0.83 TSHR (0.50) ARPGRESR2TSHRLMNA
SCHEMBL5756 0.83
Ammonia Solution, Strong SCHEMBL5912996 0.81 ESR2 (0.48) ARPGRESR2TSHRLMNA
Ammonia Solution, Strong SCHEMBL5912983 0.81 ESR2 (0.48) ARPGRESR2TSHRLMNA
SCHEMBL31655519 0.81 ESR2 (0.48) ARPGRESR2TSHRLMNA
SCHEMBL31655518 0.81 ESR2 (0.48) ARPGRESR2TSHRLMNA
SCHEMBL31366240 0.81 ESR2 (0.48) ARPGRESR2TSHRLMNA
Hydrochloric Acid SCHEMBL29026049 0.81 ESR2 (0.48) ARPGRESR2TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104136435-B bromodomain inhibitors 艾伯维公司 2017-05-10 CN disclosed