SCHEMBL28844478

SCHEMBL28844478

COc1ccc2c(C(=O)Nc3ccc(OC)c(OC)c3)cc(-c3ccccc3)nc2c1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 5/20 0.80
CYP3A4 P08684 3/20 0.72
MEN1 O00255 8/20 0.65
KMT2A Q03164 8/20 0.65
KDM4E B2RXH2 3/20 0.64
MAPT P10636 3/20 0.64
RAB9A P51151 2/20 0.63
NPC1 O15118 1/20 0.63
POLB P06746 3/20 0.62
ALDH1A1 P00352 2/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
CYP2C9 P11712 1/20 0.62
CYP2C19 P33261 1/20 0.62
CA12 O43570 3/20 0.61
CA1 P00915 3/20 0.61
CA2 P00918 3/20 0.61
CA9 Q16790 3/20 0.61
USP2 O75604 1/20 0.61
TP53 P04637 1/20 0.61
PKM P14618 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29864830 1.00 TACR3 (0.80) TACR3CYP3A4MEN1KMT2AKDM4E
SCHEMBL28844487 0.89 TACR3 (0.91) TACR3CYP3A4MEN1KMT2AKDM4E
SCHEMBL6451537 0.89 TACR3 (1.00) TACR3CYP3A4MEN1KMT2ARAB9A
SCHEMBL28844492 0.87 TACR3 (0.79) TACR3CYP3A4MEN1KMT2AMAPT
SCHEMBL29864900 0.87 TACR3 (0.79) TACR3CYP3A4MEN1KMT2AMAPT
SCHEMBL28844489 0.87 TACR3 (0.86) TACR3CYP3A4MEN1KMT2AMAPT
SCHEMBL28844493 0.87 TACR3 (0.86) TACR3CYP3A4MEN1KMT2AKDM4E
SCHEMBL28844483 0.87 TACR3 (0.86) TACR3CYP3A4MEN1KMT2AKDM4E
SCHEMBL28844490 0.85 TACR3 (0.82) TACR3CYP3A4MEN1KMT2AKDM4E
SCHEMBL28844481 0.85 TACR3 (0.82) TACR3CYP3A4MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110105279-B Quinoline STAT3 specific inhibitor and preparation method and application thereof 中山大学 2022-09-16 CN disclosed