SCHEMBL28844916

SCHEMBL28844916

CCCCN1CCCC[C@H]1C(=O)Nc1c(C)csc1C

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.73
CYP2D6 P10635 2/20 0.73
KCNH2 Q12809 1/20 0.73
POLB P06746 1/20 0.70
TSHR P16473 1/20 0.70
SMN1; SMN2 Q16637 1/20 0.70
NR1I2 O75469 1/20 0.66
KCNK3 O14649 1/20 0.64
LMNA P02545 1/20 0.64
HTT P42858 1/20 0.50
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.39
SLC6A1 P30531 1/20 0.39
CNR1 P21554 4/20 0.38
CNR2 P34972 4/20 0.38
SCN1A P35498 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN3A Q9NY46 1/20 0.38
FABP4 P15090 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28844918 1.00 CYP3A4 (0.73) CYP3A4CYP2D6KCNH2POLBTSHR
Hydrochloric Acid SCHEMBL28149111 0.99 CYP3A4 (0.76) CYP3A4CYP2D6KCNH2POLBTSHR
Hydrochloric Acid SCHEMBL28149115 0.99 CYP3A4 (0.76) CYP3A4CYP2D6KCNH2POLBTSHR
SCHEMBL28149132 0.93 KCNK3 (0.74) CYP3A4CYP2D6KCNH2POLBTSHR
SCHEMBL28149173 0.93 KCNK3 (0.74) CYP3A4CYP2D6KCNH2POLBTSHR
SCHEMBL28149134 0.93 KCNK3 (0.74) CYP3A4CYP2D6KCNH2POLBTSHR
Hydrochloric Acid SCHEMBL28149152 0.92 KCNK3 (0.72) CYP3A4CYP2D6KCNH2POLBTSHR
Hydrochloric Acid SCHEMBL28148080 0.92 KCNK3 (0.72) CYP3A4CYP2D6KCNH2POLBTSHR
Hydrochloric Acid SCHEMBL28148081 0.92 KCNK3 (0.72) CYP3A4CYP2D6KCNH2POLBTSHR
SCHEMBL28148035 0.90 CYP3A4 (0.59) CYP3A4CYP2D6KCNH2POLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106699744-B Heterocyclic amide derivative, preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2021-05-11 CN disclosed
CN-106699744-A Heterocyclic acylamide derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2017-05-24 CN disclosed