Dimethyl Maleate

Dimethyl Maleate

SCHEMBL28846293

C=C(CC(=O)OCC)C(=O)OCC.COC(=O)/C=C\C(=O)OC

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KEAP1

The experimentally established mechanism targets of Dimethyl Maleate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 known ✓ Q14145 1/20 0.45
GAA P10253 2/20 0.47
MGAM O43451 1/20 0.47
SI P14410 1/20 0.47
MGAM2 Q2M2H8 1/20 0.47
HCAR2 Q8TDS4 3/20 0.45
NFE2L2 Q16236 1/20 0.45
NPSR1 Q6W5P4 1/20 0.39
ALDH1A1 P00352 6/20 0.38
TSHR P16473 1/20 0.38
CYP2D6 P10635 2/20 0.35
CYP2C19 P33261 1/20 0.35
TRPA1 O75762 1/20 0.35
GLO1 Q04760 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33
DHODH Q02127 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL60515 0.87 GAA (0.61) GAAMGAMSIMGAM2NPSR1
Dimethyl Maleate SCHEMBL28846294 0.86 HCAR2 (0.45) HCAR2KEAP1NFE2L2NPSR1ALDH1A1
Hydrochloric Acid SCHEMBL10882428 0.85 GAA (0.58) GAAMGAMSIMGAM2NPSR1
SCHEMBL28878625 0.85 GAA (0.58) GAAMGAMSIMGAM2NPSR1
Fumaric Acid SCHEMBL28245616 0.84 HCAR2 (0.50) GAAMGAMSIMGAM2HCAR2
SCHEMBL2024186 0.82 GAA (0.50) GAAMGAMSIMGAM2NPSR1
SCHEMBL5276345 0.81 GAA (0.58) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL1597247 0.81 MGAM (0.46) GAAMGAMSIMGAM2NPSR1
SCHEMBL27862456 0.81 GAA (0.48) GAAMGAMSIMGAM2NPSR1
SCHEMBL9646080 0.80 HCAR2 (0.50) GAAMGAMSIMGAM2HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106715493-A Modified polyvinyl alcohol and water-soluble film 株式会社可乐丽 2017-05-24 CN disclosed