SCHEMBL2884665

SCHEMBL2884665

O=C(O)c1ccc(C(=O)c2cc[c]cc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 12/20 0.71
TSHR P16473 3/20 0.57
TP53 P04637 1/20 0.57
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA12 O43570 1/20 0.48
CA3 P07451 1/20 0.48
TYR P14679 1/20 0.48
DRD1 P21728 1/20 0.48
CA4 P22748 1/20 0.48
CA6 P23280 1/20 0.48
CA5A P35218 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48
CA5B Q9Y2D0 1/20 0.48
ALDH1A1 P00352 2/20 0.46
ALOX15 P16050 1/20 0.46
TPMT P51580 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8070391 0.90 TSHR (0.61) SRD5A2TSHRTP53CA1CA2
SCHEMBL20583 0.90
SCHEMBL28987694 0.87 TSHR (0.58) SRD5A2TSHRTP53CA1CA2
SCHEMBL27838461 0.87 TSHR (0.58) SRD5A2TSHRTP53CA1CA2
SCHEMBL28182301 0.87 TSHR (0.58) SRD5A2TSHRTP53CA1CA2
SCHEMBL28642392 0.87 TSHR (0.58) SRD5A2TSHRTP53CA1CA2
SCHEMBL7571173 0.87 TSHR (0.58) SRD5A2TSHRTP53CA1CA2
SCHEMBL29124318 0.87 TSHR (0.58) SRD5A2TSHRTP53CA1CA2
SCHEMBL27474165 0.87 TSHR (0.58) SRD5A2TSHRTP53CA1CA2
SCHEMBL27887947 0.87 TSHR (0.58) SRD5A2TSHRTP53CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3334767-A1 PHOTOACTIVATABLE FOULING-RESISTANT COPOLYMERS Arrow International, Inc. (US) 2018-06-20 EP disclosed
WO-2017030950-A1 PHOTOACTIVATABLE FOULING-RESISTANT COPOLYMERS ARROW INTERNATIONAL, INC. (US) 2017-02-23 WO disclosed
US-7776893-B2 Use of PDE4 inhibitors for the treatment of diabetes mellitus NYCOMED GMBH (DE) 2010-08-17 US disclosed
US-20060281745-A1 Use of pde4 inhibitors for the treatment of diabetes mellitus ALTANA PHARMA AG (DE) 2006-12-14 US disclosed
EP-1650193-A2 6-Phenylphenanthridines with PDE-IV inhibiting activity ALTANA Pharma AG (DE) 2006-04-26 EP disclosed
EP-1147089-B1 PHENYLPHENANTHRIDINES WITH PDE-IV INHIBITING ACTIVITY ALTANA PHARMA AG (DE) 2005-12-07 EP disclosed
CN-1152864-C Phenylphenanthridines with PDE-IV inhibiting activity ��̹��ҽҩ��˾ 2004-06-09 CN disclosed
US-6476025-B1 Phenylphennanthridines with PDE-IV inhibiting activity ALTANA PHARMA AG (DE) 2002-11-05 US disclosed
CN-1336919-A Phenylphenanthridines with PDE-IV inhibiting activity BYK GULDEN LOMBERG CHEM FAB (DE) 2002-02-20 CN disclosed
EP-1147089-A1 PHENYLPHENANTHRIDINES WITH PDE-IV INHIBITING ACTIVITY Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 2001-10-24 EP disclosed
WO-2000042020-A1 PHENYLPHENANTHRIDINES WITH PDE-IV INHIBITING ACTIVITY BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-07-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060281745-A1 Use of pde4 inhibitors for the treatment of diabetes mellitus PDE4A, PDE4B, PDE12 SRD5A2 434/4885TSHR 3470/4885TP53 4341/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.