SCHEMBL28851111

SCHEMBL28851111

Cc1ccc(Br)c(CO[Si](C)(C)C(C)(C)C)n1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.33
USP2 O75604 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ALDH1A1 P00352 2/20 0.33
GFER P55789 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29664278 1.00 KDM4E (0.33) KDM4EUSP2HPGDHSD17B10ALDH1A1
SCHEMBL23089668 0.86 CA12 (0.31)
SCHEMBL18836819 0.81 PREP (0.31)
SCHEMBL694083 0.81 KDM4E (0.51) KDM4EUSP2HPGDHSD17B10ALDH1A1
SCHEMBL28850991 0.80 TACR1 (0.34)
SCHEMBL29689720 0.80 TACR1 (0.34)
SCHEMBL29080416 0.78 KDM4E (0.35) KDM4EHPGDALDH1A1
SCHEMBL29978430 0.77 CYP1A2 (0.46) KDM4EALDH1A1
SCHEMBL610829 0.76 TACR1 (0.37) KDM4EHPGDALDH1A1
SCHEMBL18322436 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114127073-B Imidazopyrimidines as EED inhibitors and use thereof 密歇根大学董事会 2024-05-31 CN disclosed
CN-115212311-A Pharmaceutical composition and application thereof 苏州亚盛药业有限公司 2022-10-21 CN disclosed
CN-114127073-A Imidazopyrimidines as EED inhibitors and uses thereof 美国密歇根州立大学试剂中心 2022-03-01 CN disclosed