SCHEMBL28855733

SCHEMBL28855733

CCC(=O)N1C[C@H](Nc2ncnc3[nH]ccc23)CC[C@@H]1C

nearest known ligand 0.73

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 19/20 0.73
JAK1 P23458 3/20 0.73
BTK Q06187 2/20 0.73
TEC P42680 1/20 0.73
TXK P42681 1/20 0.73
BLK P51451 1/20 0.73
BMX P51813 1/20 0.73
ITK Q08881 1/20 0.73
ERBB4 Q15303 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24106806 0.90 BTK (0.71) JAK3JAK1BTKTECTXK
SCHEMBL24867427 0.88 JAK3 (0.77) JAK3JAK1BTKTECTXK
SCHEMBL26095750 0.88 JAK3 (0.77) JAK3JAK1BTKTECTXK
Ritlecitinib SCHEMBL16785968 0.84 JAK3 (1.00) JAK3JAK1BTKTECTXK
Ritlecitinib SCHEMBL22511885 0.84 JAK3 (1.00) JAK3JAK1BTKTECTXK
Ritlecitinib SCHEMBL16765061 0.84 JAK3 (1.00) JAK3JAK1BTKTECTXK
Ritlecitinib SCHEMBL19595622 0.84 JAK3 (1.00) JAK3JAK1BTKTECTXK
Ritlecitinib SCHEMBL16764793 0.84 JAK3 (1.00) JAK3JAK1BTKTECTXK
Ritlecitinib SCHEMBL16764638 0.84 JAK3 (1.00) JAK3JAK1BTKTECTXK
Ritlecitinib SCHEMBL30208783 0.84 JAK3 (1.00) JAK3JAK1BTKTECTXK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115023221-A Stable immediate release tablet and capsule formulations of 1- ((2S,5R) -5- ((7H-pyrrolo [2,3-D ] pyrimidin-4-yl) amino) -2-methylpiperidin-1-yl) prop-2-en-1-one 辉瑞英国研发有限公司 2022-09-06 CN disclosed