SCHEMBL28859836

SCHEMBL28859836

CC1(C)Cc2ccccc2N(c2ccccc2)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.43
TMEM97 Q5BJF2 4/20 0.43
HTR7 P34969 3/20 0.43
HTR2B P41595 3/20 0.43
SLC6A2 P23975 3/20 0.43
HTR1A P08908 2/20 0.43
ADRA2A P08913 2/20 0.43
ADRA2B P18089 2/20 0.43
ADRB3 P13945 1/20 0.43
DRD4 P21917 1/20 0.43
HTR2C P28335 1/20 0.43
ADRA1A P35348 1/20 0.43
SLC6A3 Q01959 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
ADRA2C P18825 2/20 0.42
ADRB1 P08588 1/20 0.42
HRH2 P25021 1/20 0.42
ADRA1D P25100 1/20 0.42
NOTUM Q6P988 1/20 0.38
MTNR1A P48039 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16687886 0.76 NOTUM (0.41) HTR7HTR2BHTR1AHTR2CNOTUM
SCHEMBL21662887 0.74 NOTUM (0.33) NOTUMHPGDNPC1RAB9ALMNA
SCHEMBL20088333 0.74 NOTUM (0.35) SIGMAR1HTR2BHTR2CADRA2CNOTUM
SCHEMBL23561017 0.74 GRM5 (0.54) SIGMAR1TMEM97NPC1RAB9ASMN1; SMN2
SCHEMBL7262697 0.74 NOTUM (0.40) HTR7HTR2BSLC6A2HTR1AHTR2C
SCHEMBL13647676 0.71 NOTUM (0.38) SLC6A2NOTUMHPGDSMN1; SMN2ALDH1A1
SCHEMBL2625757 0.71 NOTUM (0.38) SLC6A2HTR1AADRA2AADRA1ASLC6A3
SCHEMBL8013849 0.71 TMEM97 (0.40) SIGMAR1TMEM97HTR7HTR2BSLC6A2
SCHEMBL3304748 0.70 NOTUM (0.50) SIGMAR1TMEM97HTR7HTR2BSLC6A2
SCHEMBL11430704 0.70 NPC1 (0.53) SIGMAR1SLC6A2ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105189461-B The dibasic 1- acyl groups -4- amino -1,2,3,4- tetrahydroquinoline derivatives of 2,3- and their purposes as bromine domain inhibitor 葛兰素史克知识产权第二有限公司 2018-05-15 CN disclosed