SCHEMBL28860458

SCHEMBL28860458

CNc1nc(Nc2ccc(N3CCOCC3)nc2)ncc1C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.54
JAK1 P23458 1/20 0.51
JAK3 P52333 1/20 0.51
JAK2 O60674 1/20 0.51
LRRK2 Q5S007 1/20 0.51
SYK P43405 5/20 0.51
IGF1R P08069 3/20 0.50
DGAT1 O75907 2/20 0.50
TBK1 Q9UHD2 1/20 0.50
CYP1A2 P05177 2/20 0.49
CSF1R P07333 1/20 0.49
DAPK1 P53355 1/20 0.49
KCNH2 Q12809 1/20 0.49
STAT6 P42226 2/20 0.48
MAPT P10636 1/20 0.48
CYP2C19 P33261 1/20 0.48
INSR P06213 1/20 0.48
PTK2 Q05397 1/20 0.48
PTK2B Q14289 1/20 0.48
PKMYT1 Q99640 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18171846 0.86 EGFR (0.50) EGFRJAK1JAK3JAK2LRRK2
SCHEMBL18181558 0.85 JAK1 (0.53) EGFRJAK1JAK3JAK2LRRK2
SCHEMBL18171849 0.82 JAK1 (0.50) EGFRJAK1JAK3JAK2LRRK2
SCHEMBL18181611 0.80 JAK1 (0.50) EGFRJAK1JAK3JAK2LRRK2
SCHEMBL20073216 0.78 JAK1 (0.49) EGFRJAK1JAK3JAK2LRRK2
SCHEMBL15358443 0.76 SYK (0.60) EGFRJAK3JAK2SYKIGF1R
SCHEMBL28221625 0.76 PLK4 (0.56) JAK1JAK3JAK2IGF1R
SCHEMBL18181563 0.75 MAPT (0.51) EGFRCYP1A2CSF1RDAPK1KCNH2
SCHEMBL15349506 0.75 SYK (0.59) EGFRJAK3JAK2SYKIGF1R
SCHEMBL468661 0.74 CYP1A2 (0.58) DGAT1CYP1A2MAPTCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137593-A PREPARATION AND USE OF NOVEL PROTEIN KINASE INHIBITORS 上海交通大学医学院附属瑞金医院 2018-06-08 CN disclosed